Testing Status of 2-Ethylhexyl p-Methoxycinnamate M20239
CASRN: 5466-77-3
Related: 2-Hydroxy-4-methoxybenzophenone
Formula: C18-H26-O3
Synonyms/Common Names
- EHMC
- 2-Ethylhexyl methoxycinnamate
- Octinoxate
- 2-Propenoic acid, 3-(4-methoxyphenyl)-, 2-ethylhexyl ester (9CI)
Modified One-Generation
- GD 6 to PND 28 Dose Range Finding (Dosed-Feed)
(MOG003)
Completed
- Citation: National Toxicology Program (NTP). 2022. NTP developmental and reproductive toxicity technical report on the modified one-generation study of 2-ethylhexyl p methoxycinnamate (CASRN 5466-77-3) administered in feed to Sprague Dawley (Hsd:Sprague Dawley SD) rats with prenatal, reproductive performance, and subchronic assessments in F1 offspring. Research Triangle Park, NC: National Toxicology Program. DART Report 06. https://doi.org/10.22427/NTP-DART-06
- Female Rats: Harlan Sprague-Dawley
- Dose: 0, 2250, 5000, 10,000 or 20,000 ppm.
- Developmental Toxicity (Dosed-Feed)
(MOG003B)
Completed
- Prenatal Developmental Toxicity
- Citation: National Toxicology Program (NTP). 2022. NTP developmental and reproductive toxicity technical report on the modified one-generation study of 2-ethylhexyl p methoxycinnamate (CASRN 5466-77-3) administered in feed to Sprague Dawley (Hsd:Sprague Dawley SD) rats with prenatal, reproductive performance, and subchronic assessments in F1 offspring. Research Triangle Park, NC: National Toxicology Program. DART Report 06. https://doi.org/10.22427/NTP-DART-06
- Rats: Harlan Sprague-Dawley
- Dose: 0, 1000, 3000, or 6000 ppm.
- F0 Generation (Dosed-Feed)
(MOG003B)
Completed
- F0 Generation
- Citation: National Toxicology Program (NTP). 2022. NTP developmental and reproductive toxicity technical report on the modified one-generation study of 2-ethylhexyl p methoxycinnamate (CASRN 5466-77-3) administered in feed to Sprague Dawley (Hsd:Sprague Dawley SD) rats with prenatal, reproductive performance, and subchronic assessments in F1 offspring. Research Triangle Park, NC: National Toxicology Program. DART Report 06. https://doi.org/10.22427/NTP-DART-06
- Rats: Harlan Sprague-Dawley
- Fertility Assessment (Dosed-Feed)
(MOG003B)
Completed
- Fertility Assessment
- Citation: National Toxicology Program (NTP). 2022. NTP developmental and reproductive toxicity technical report on the modified one-generation study of 2-ethylhexyl p methoxycinnamate (CASRN 5466-77-3) administered in feed to Sprague Dawley (Hsd:Sprague Dawley SD) rats with prenatal, reproductive performance, and subchronic assessments in F1 offspring. Research Triangle Park, NC: National Toxicology Program. DART Report 06. https://doi.org/10.22427/NTP-DART-06
- Rats: Harlan Sprague-Dawley
- Dose: 0, 1000, 3000, or 6000 ppm.
- 13-Week Subchronic (Dosed-Feed)
(MOG003B)
Completed
- Citation: National Toxicology Program (NTP). 2022. NTP developmental and reproductive toxicity technical report on the modified one-generation study of 2-ethylhexyl p methoxycinnamate (CASRN 5466-77-3) administered in feed to Sprague Dawley (Hsd:Sprague Dawley SD) rats with prenatal, reproductive performance, and subchronic assessments in F1 offspring. Research Triangle Park, NC: National Toxicology Program. DART Report 06. https://doi.org/10.22427/NTP-DART-06
- Rats: Harlan Sprague-Dawley
- Dose: 0, 1000, 3000, or 6000 ppm.
Special Studies
- Absorption Distribution Metabolism Excretion (Dermal; Intravenous; Gavage; Dermal; Intravenous; Gavage)
(K20239)
Completed
- Citation: Fennell TR, Mathews JM, Snyder RW, Hong Y, Watson SL, Black SR, McIntyre BS, Waidyanatha S. Metabolism and disposition of 2-ethylhexyl-p-methoxycinnamate following oral gavage and dermal exposure in Harlan Sprague Dawley rats and B6C3F1/N mice and in hepatocytes in vitro. Xenobiotica. 2018 Nov;48(11):1142-1156. doi: 10.1080/00498254.2017.1400129. Epub 2017 Nov 23.Pubmed Abstract
- Male and Female Rats: Harlan Sprague-Dawley; Male and Female Mice: B6C3F1
- Dose: 0.8, 8, 80 mg/kg [R,M]. 8 mg/kg. 8 mg/kg [R,M]. 8, 80, 800 mg/kg.
- 3 days Hershberger Assay (Gavage)
(K20239D)
Completed
- Citation: National Toxicology Program (NTP). 2020. NTP technical report on the toxicology and carcinogenesis studies of 2-hydroxy-4-methoxybenzophenone (CASRN 131-57-7) administered in feed to Sprague Dawley (Hsd:Sprague Dawley SD) rats and B6C3F1/N mice. Research Triangle Park, NC: National Toxicology Program. Technical Report 597. https://doi.org/10.22427/NTP-TR-597
- Male Rats: Harlan Sprague-Dawley
- Dose: 0, 100, 320, 1000 mg/kg.
- Preliminary Toxicokinetic Study (Dosed-Feed; Gavage; Intravenous)
(K20239E)
Completed
- Male and Female Rats: Harlan Sprague-Dawley
- Dose: 20,000 ppm. 8 mg/kg. 80, 800 mg/kg.
- 3 days Uterotrophic Assay (Gavage)
(K20239C)
Completed
- Citation: National Toxicology Program (NTP). 2020. NTP technical report on the toxicology and carcinogenesis studies of 2-hydroxy-4-methoxybenzophenone (CASRN 131-57-7) administered in feed to Sprague Dawley (Hsd:Sprague Dawley SD) rats and B6C3F1/N mice. Research Triangle Park, NC: National Toxicology Program. Technical Report 597. https://doi.org/10.22427/NTP-TR-597
- Female Rats: Sprague Dawley
- Dose: 0, 320, 1000 mg/kg.
Genetic Toxicology
- Micronucleus
(G20239B)
Completed
- Rats: Harlan Sprague-Dawley
- Male Negative
- Female Negative
- Salmonella
(201557)
Completed
- Citation: Zeiger, E., Haworth, S., Mortelmans, K., and Speck, W. Mutagenicity testing of Di(2-ethylhexyl)phthalate and related chemicals in Salmonella Environ. Mutagen. Vol. 7 (1985) 213-232
- Negative
- Salmonella
(G20239)
Completed
- Negative
Organ Systems Toxicity
- varies Immunotoxicity (Topical Application)
(I20239)
Completed
- Female Mice: BALB/c
- Dose: 0, 2.5%, 5.0%, 10%, 25%, 50%.
in vitro Testing
- H295R Steroidogenesis Assay
(V20239)
Completed
- H295R Steroidogenesis Assay
- Human (Cell Lines)
- Androgen Receptor Binding Assay
(V20239B)
Completed
- Androgen receptor Binding Assay
- Rats: Sprague Dawley
- Estrogen Receptor Binding Assay
(V20239C)
Completed
- Estrogen Receptor Binding Assay
- Rats: Sprague Dawley
- Androgen Receptor Transactivation Assay
(V20239D)
Completed
- Androgen Receptor Transactivation Assay
- Human (Cell Lines)
- Estrogen Receptor Transactivation Assay
(V20239E)
Completed
- Estrogen Receptor Transactivation Assay
- Human (Cell Lines)
- Human Recombinant Aromatase Assay
(V20239G)
Completed
- Human Recombinant Aromatase Assay
- Human (Cell Lines)